Mgbakwunye akwara mgbochi Estrogen Steroid White ntụ ntụ Tamoxifen Citrate Nolvadex
Ngwa ngwa nkọwa
Ngwaahịa: Nolvadex (Tamoxifen Citrate)
Nọmba CAS: 54965-24-1
MF: C26H29NO
MW: 371.51
Dị ọcha: 99%
Ebe esi mmiri: 482.3°C na 760 mmHg
Nchekwa: Akara akara na 2 ºC -8 ºC
Ebe mgbaze: 140-144 Celsius
ọkụ ọkụ: 356.5ºC
Nhazi:
Nọmba Einecs: 234-118-0
Ọkọlọtọ: Standard Enterprise
Ngwaahịa mgbochi ọrịa cancer ndị ọzọ: Tamoxifen Citrate, Clomiphene Citrate, Toremifene Citrate, Anastrozole, Raloxifene hydrochloride, Fulvestrant, Letrozole, Crotamiton
Ojiji:Tamoxifen bụ homonụ nwanyị nke nwere ike igbochi omume estrogen, a na-ejikarị ya agwọ ụdị ọrịa ara ara na nwoke na nwanyị.
Steroid ọgwụgwọ ọrịa kansa anyị na-enye
Tamoxifen Citrate | onye na-abụghị steroidal |
Exemestane | ihe mgbochi aromatase |
Anastrozole | eji eme ihe mgbe ị na-eji nnukwu ihe na-esi ísì ụtọ |
Stanozolol | Ịcha okirikiri |
Toremifene Citrate | Estrogen receptor modulator na-abụghị steroidal nhọrọ |
Drostanolone Propionate | Steroid anabolic |
Methenolone Enanthate | na protein homonụ assimilation ike ọrụ nke imeju |
17-methyltestosterone | Androgen na Albumen Assimilation steroid |
Fluoxymesterone | enwere ike iji ya mee ihe dị ka ọgwụ ọgwụ |
Formestan | A na-eji ya dị ka ihe mgbochi enzyme aromatic |
Ntụziaka Nolvadex
ntụ ntụ: kwa 1 gram nke Tamoxifen citrate
Na-emepụta: ntinye kachasị elu mere - 20 mg / ml
Ihe achọrọ:
1 gram nke Tamoxifen Citrate
1 beaker kwesịrị ekwesị maka ijide olu nke mmiri mmiri
19.6 ml nke glycerol
29.4 ml nke mmanya mmanya na-egosi ọka 190
ntụ ntụ: kwa 1 gram nke Tamoxifen citrate
Na-emepụta: ntinye kachasị elu mere - 20 mg / ml
Ihe achọrọ:
1 gram nke Tamoxifen Citrate
1 beaker kwesịrị ekwesị maka ijide olu nke mmiri mmiri
9.8 ml nke PEG 600
39.2 ml nke mmanya mmanya na-egosi ọka 190
Nolvadex ojiji na usoro onunu ogwu
Ọrịa ara ara | 10 ka 20 mg ọnụ ugboro abụọ kwa ụbọchị |
Maka ọrịa kansa metastatic | 20 ruo 40 mg nyere na nkewa |
Ụmụ nwanyị nwere Ductal Carcinoma | 20 mg kwa ụbọchị maka afọ 5 |
Belata ọrịa kansa ara | 20mg kwa ụbọchị maka afọ 5 |
Node-positive cancer ara, axillary dissection | 10 mg ọnụ 2 ruo 3 ugboro kwa ụbọchị maka afọ 5. |
Ụmụ agbọghọ dị afọ 2 ruo 10 nwere ọrịa McCune-Albright | 20 mg kwa ụbọchị maka otu afọ |
Ngwa Nolvadex
1: Tamoxifen Citrate Jiri na Cancer
Tamoxifen citrate | Ekwenyere iji gbochie: Ọrịa ara ara na ụmụ nwanyị ndị nwere nnukwu ihe ize ndụ maka ọrịa ahụ. |
Ọrịa ara ara na ụmụ nwanyị na ụmụ nwoke | |
a na-amụ na ọgwụgwọ ụdị ọrịa cancer ndị ọzọ. |
2: Uru nke Tamoxifen
A. Tamoxifen na-ebelata ma ọ bụ kwụsị uto mkpụrụ ndụ kansa nke dịlarị n'ime ahụ.Ọ na-enyere aka mee ka ọrịa cancer ara mbụ ghara ịlọghachi ma na-enyere aka igbochi ọrịa cancer ọhụrụ na ara na-abụghị.Ọ na-ebelatakwa ohere nke ọrịa kansa ara na ụmụ nwanyị nwere nnukwu ihe ize ndụ maka ọrịa a.
B. A na-eji Tamoxifen egbochi ma na-agwọ ọrịa cancer ara nke na-anwale ihe dị mma maka ndị na-anabata estrogen (ER +).Ọ na-egbochi mmetụta nke estrogen hormone nwere na mkpụrụ ndụ kansa ma na-ebelata ohere nke ọrịa ara ara ga-eto eto.A na-akpọkarị ya "anti-estrogen."
C. Tamoxifen na-arụ ọrụ nke ọma n'ibelata ihe ize ndụ nke nlọghachi ọrịa kansa ara.N'ime ụmụ nwanyị ndị nwere ọrịa ara ara, tamoxifen na-ebelata ohere nke ọrịa ara ara na ara na-abụghị (contralateral)
D. Maka ụmụ nwanyị postmenopausal, ọgwụgwọ nke abụọ na-eji tamoxifen wee bụrụ ihe mgbochi aromatase, dị ka anastrozole (Arimidex), exemestane (Aromasin), ma ọ bụ letrozole (Femara) nwere ike ịrụ ọrụ nke ọma karịa naanị ịta tamoxifen.